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24-well plate:

1 A1 Tre:BACE2+FRET Substrate 2 0 Dox2 A2 Tre:miRG1,Hef1a:BACE1 (0 Dox) +FRET Substrate 13 A3 Tre:miRG1,Hef1a:BACE1 (1000 Dox) +FRET Substrate 14 A4 Tre:BACE2+FRET Substrate 2 1000 Dox5 A5 Assay Buffer 1 + FRET Substrate 16 A6 Assay Buffer 2 + FRET Substrate 2
13 B1 5 uM Reference Standard+ FRET 114 B2 2.5 uM Reference Standard+ FRET 115 B3 1.25 uM Reference Standard+ FRET 116 B4 0.63 uM Reference Standard+ FRET 117 B5 0.32 uM Reference Standard+ FRET 118 B6 0.16 uM Reference Standard+ FRET 1
19 C1 5 uM Reference Standard+ FRET 220 C2 2.5 uM Reference Standard+ FRET 221 C3 1.25 uM Reference Standard+ FRET 222 C4 0.63 uM Reference Standard+ FRET 223 C5 0.32 uM Reference Standard+ FRET 224 C6 0.16 uM Reference Standard+ FRET 2

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